5
Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T14776 | BRD4 Inhibitor-10 | Epigenetic Reader Domain | |
BRD4 Inhibitor-10 is an inhibitor of BRD4-BD1 (IC50: 8 nM). | |||
T1854 | MS436 | Epigenetic Reader Domain | |
MS436 is a selective, small-molecule inhibitor for the BRD4 bromodomains. | |||
T61387 | Bromodomain inhibitor-10 | ||
Bromodomain inhibitor-10 (compound 128) is a highly potent inhibitor of bromodomain activity. It exhibits strong binding affinity with K d values of 15.0 nM and 2500 nM for BRD4-1 and BRD4-2, respectively. Furthermore, B... | |||
T36103 | TW9 | TW9 | |
TW9 is a dual inhibitor of bromodomain 2 (BD2) in bromodomain-containing protein 4 (BRD4) and histone deacetylase 1 (HDAC1; IC50s = 0.074 and 0.29 μM, respectively).1It is selective for BD2 over BD1 in BRD4 (IC50= 0.72 μ... | |||
T38381 | CAY17c | ||
CAY17c is an inhibitor of bromodomain-containing protein 4 (BRD4; IC50= 0.71 μM), as well as class I histone deacetylases (HDACs; IC50s = 0.046, 0.058, 0.075, and 0.167 μM for HDAC1, -2, -3, and -8, respectively) and cla... |